Publications
Clinical Publications
2022
A Randomized, Factorial Phase II Study to Determine the Optimal Dosing Regimen for 68Ga-Satoreotode Trizoxetan as an Imging Agent in Patients with Gastroenteropancreatic Neuroendocrine Tumors.
Virgolini I et al.
J Nucl Med 2022; 63: 376-383.
2021
A novel read methodology to evaluate the optimal dose of 68Ga-satoreotide trizoxetan as a PET imaging agent in pts with gastroenteropancreatic neuroendocrine tumours: a phase II clinical trial.
Miller CG et al.
EJNMMI Res 2021; 11: 84.
Safety and Effectiveness of 177Lu-Satoreotide Tetraxetan in Patients with Progressive Neuroendocrine Tumors (NETs): Interim Analysis of a Phase I/II Study.
Grønbæk H et al.
NANETS 2021, C-31: Poster 411.
2019
Phase I Trial of Well-Differentiated Neuroendocrine Tumors (NETs) with Radiolabeled Somatostatin Antagonist 177Lu-Satoreotide Tetraxetan.
Reidy-Lagunes D et al.
Clin Cancer Res 2019; 25(23):6939-6947.
2018
Safety, Biodistribution, and Radiation Dosimetry of 68Ga-OPS202 in patients with Gastroenteropancreatic Neuroendocrine Tumors: A Prospective Phase I Imaging Study.
Nicolas GP et al.
J Nucl Med 2018; 59: 909-914.
Sensitivity Comparison of 68Ga-OPS202 and 68Ga-DOTATOC PET/CT in patients with Gastroenteropancreatic Neuroendocrine Tumors: A Prospective Phase II Imaging Study.
Nicolas GP et al.
J Nucl Med 2018; 59: 915-921.
2014
Comparison of Somatostatin Receptor Agonist and Antagonist for Peptide Receptor Radionuclide Therapy: A Pilot Study.
Wild D et al.
J Nucl Med 2014; 55(8): 1248-1252.
Non-clinical Publications
2021
Distinct In Vitro Bindong Profile of the Somatostatin Receptor Subtype 2 Antagonist [177Lu]Lu-OPS201 Compared to the Agonist [177Lu]Lu-DOTA-TATE.
Mansi R et al.
Pharmaceuticals 2021; 14: 1265.
2019
Design and development of the theranostic pair 177Lu-OPS201/68Ga-OPS202 for targeting somatostatin receptor expressing tumors.
Mansi R et al.
J Labelled Compounds RPs 2019; 62(10): 635-645.
2017
Somatostatin Receptor Antagonists for Imaging and Therapy.
Fani M et al.
J Nucl Med 2017; 58: 61S-66S.
2016
Comparison of the Therapeutic Response to Treatment with a 177Lu-Labeled SSTR Agonist and Antagonist in Preclinical Models.
Dalm SU et al.
J Nucl Med 2016; 57: 260-265.
2011
PET of Somatostatin Receptor-Positive Tumors Using 64Cu- and 68Ga-Somatostatin Antagonoists: The Chellate Makes the Difference.
Fani M et al.
J Nucl Med 2011; 52: 1110-1118.
2008
Design and in vitro Characterization of Highly Sst2-selective Somatostatin Antagonists Suitable for Radio-Targeting.
Cescato R et al.
J Med Chem 2008; 51-13:4030-4037.
2006
Radiolabeled somatostatin antagonists are preferable to agonists for in vivo peptide receptor targeting of tumors.
Ginj M et al.
PNAS 2006; 103(44): 16436-16441.
© Ariceum Therapeutics
